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1. diaConjugation of salicylic acid 16.bin morphin steroids Dubin Johnson syndr. Ways of conjugation Sulfation – PAPS - sulfotransferases Sulfation – PAPS –

Slide 1BIOTRANSFORMATION, Drug metabolism, detoxification Phase 2 conjugation Slide 2 su sulfation Glucuronidation (80%) Conjugation with amino acids glycosylation acetylation…

Francesco Regoli Detoxification and biotransformation of xenobiotics in marine organisms Department of Life and Environmental Sciences Polytechnic University of Marche-Ancona…

PHARMACOKINETICS PHARMACOKINETICS BIOTRANSFORMATION Drug metabolism/drug inactivation/drug detoxification The chemical alteration of drug molecules by the body cells of patients…

1.Dr. Rahul Kunkulol , Asso. professor, Dept. Of Pharmacology 2. • The chemical modification of drugs with the overall goal of getting rid of the drug • Enzymes are typically…

Biotransformation Xenobiotic metabolism “Essentials of Toxicology” by Klaassen Curtis D. and Watkins John B Chapter 6 Biotransformation Water soluble xenobiotics are…

Biotransformation BIOTRANSFORMATION Dr.RENJU.S.RAVI MD OVERVIEW Definition Consequences Types Phase I/II in detail Enzyme Induction/Inhibition First Pass Metabolism Xenobiotics-…

Biotransformation BIOTRANSFORMATION Dr.RENJU.S.RAVI MD OVERVIEW Definition Consequences Types Phase I/II in detail Enzyme Induction/Inhibition First Pass Metabolism Xenobiotics-…

Functional Medicine University’s Functional Diagnostic Medicine Training Program Module 6 * FMDT 551A The Physiology and Biochemistry of Biotransformation/Detoxification…

PHARMACOKINETICS Part 3 BIOTRANSFORMATION Drug metabolism/drug inactivation/drug detoxification The chemical alteration of drug molecules by the body cells of patients to…

1. Biotransformation(Metabolism) of Drugs 2. A. General properties1. Biotransformation is a major mechanism for drug elimination;• Results of biotransformation: – Production…

8172019 CS_K18 Drug Metabolism - Biotransformation 132 DRUG METABOLISM BIOTRANSFORMA TIONAznan Lelo Yunita Sari Pane De! Fara#olo$i %an Teraeuti# Fa#ulta e%o#teran…

PowerPointhydrolysis) Several routes of metabolism found in vivo May inactivate or bioactivate action Liver is the major site of metabolism Genetically variation with some

The Detoxification System Part II: Hepatic Biotransformation by Mark J Donohue Introduction By the early 21st century our society has increasingly been exposed to more and…

Drug Metabolism By: Dr Mohsen Bebars Dr Mohsen Bebars Drug Metabolism Biotransformation ➢ It is a process of biochemical changes of drugs or xenobiotics in the body which…

Vol 55 No 1APPLIED AND ENVIRONMENTAL MICROBIOLOGY Jan 1989 p 190-197 0099-224089010190-08$02000 Copyright © 1989 American Society for Microbiology Biotransformation and…

CS_avhandling_reprosentralen_korrekt_versjon.pdfin rats and Ahr knockout mice Dissertation for the degree of Ph.D. by National Institute of Occupational Health, Oslo, Norway

Metabolic Transformations of Xenobiotics Introduction of Biotransformation reactions Amin M. Kamel, Ph.D. Pfizer Global Research and Development Groton Laboratories Bioanalytical…

Slide 1 DR.SOBAN SADIQ Slide 2 Pharmacokinetics Absorption Distribution Metabolism(Biotransformation) Excretion Slide 3 Slide 4 Routes of drug administration Enteral(Through…

Metabolism of xenobiotics FM 3.5-10 CHE 5-6 Metabolism of xenobiotics Also called: ! Biotransformation, or detoxification Primary metabolism – secondary metabolism Goal:…