ChemInform Abstract: Synthesis of 4-Aryl-4,5-dihydro-1H-indeno[1,2-d]pyrimidines by Biginelli...

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ChemInform 2011, 42, issue 47 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim Fused pyrimidine derivatives R 0515 DOI: 10.1002/chin.201147157 Synthesis of 4-Aryl-4,5-dihydro-1H-indeno[1,2-d]pyrimidines by Biginelli Con- densation and Their Antibacterial Activities. — A variety of new indenopyrimi- dinethiones (V) is synthesized via a multi-component condensation reaction under mi- crowave irradiation conditions. Thiones (IV) and corresponding S-alkylated/S-benzy- lated products are evaluated for their antibacterial activities. S-alkylated indenopy- rimidine derivatives (Va) and (Vb) appear to be the most potent samples. — (KAUR, R.; BANSAL, M.; KAUR*, B.; MISHRA, T.; BHATIA, A.; J. Chem. Sci. (Bangalore, India) 123 (2011) 4, 443-451 ; Dep. Chem., Punjabi Univ., Patiala 147 002, India; Eng.) — C. Cyrus 47- 157

Transcript of ChemInform Abstract: Synthesis of 4-Aryl-4,5-dihydro-1H-indeno[1,2-d]pyrimidines by Biginelli...

Page 1: ChemInform Abstract: Synthesis of 4-Aryl-4,5-dihydro-1H-indeno[1,2-d]pyrimidines by Biginelli Condensation and Their Antibacterial Activities.

Fused pyrimidine derivativesR 0515 DOI: 10.1002/chin.201147157

Synthesis of 4-Aryl-4,5-dihydro-1H-indeno[1,2-d]pyrimidines by Biginelli Con-densation and Their Antibacterial Activities. — A variety of new indenopyrimi-dinethiones (V) is synthesized via a multi-component condensation reaction under mi-crowave irradiation conditions. Thiones (IV) and corresponding S-alkylated/S-benzy-lated products are evaluated for their antibacterial activities. S-alkylated indenopy-rimidine derivatives (Va) and (Vb) appear to be the most potent samples. — (KAUR, R.; BANSAL, M.; KAUR*, B.; MISHRA, T.; BHATIA, A.; J. Chem. Sci. (Bangalore, India) 123 (2011) 4, 443-451 ; Dep. Chem., Punjabi Univ., Patiala 147 002, India; Eng.) — C. Cyrus

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ChemInform 2011, 42, issue 47 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim

MER: a shell script and annotation server for minimal named ......Couto and Lamurias J Cheminform Page 5 of 10 common,sandswesempiricallysfoundsthatsmostsofsthestwo-charactersmatchesswereserrors

MER: a shell script and annotation server for minimal named ......Couto and Lamurias J Cheminform Page 5 of 10 common,sandswesempiricallysfoundsthatsmostsofsthestwo-charactersmatchesswereserrors

Synthesis and Characterization of Novel Biginelli ...downloads.hindawi.com/journals/jchem/2019/3131879.pdf · 5-(nitro/bromo)-styryl-2-benzimidazoles derivatives and screened for

Synthesis and Characterization of Novel Biginelli ...downloads.hindawi.com/journals/jchem/2019/3131879.pdf · 5-(nitro/bromo)-styryl-2-benzimidazoles derivatives and screened for

Reação de Biginelli: uso de ácidos p-sulfônico-calix[n ...

Reação de Biginelli: uso de ácidos p-sulfônico-calix[n ...

RESEARCHARTICLE Assessingtheinformationcontent ......Rodríguez‑Pérezet al. J Cheminform Page6of14 whichyieldedmedianMCCvaluesof0.67(IFP_85) and0.63(EFCP_folded).us,inhibitorswithbinding

RESEARCHARTICLE Assessingtheinformationcontent ......Rodríguez‑Pérezet al. J Cheminform Page6of14 whichyieldedmedianMCCvaluesof0.67(IFP_85) and0.63(EFCP_folded).us,inhibitorswithbinding

RESEARCHARTICLE LargescalecomparisonofQSAR … · 2020. 3. 19. · Boscet al. J Cheminform Page3of16 Dta preparation Compoundstructureswereextractedfromthedatabase inSMILESformatandusingRDKit(version2017_09_01)

RESEARCHARTICLE LargescalecomparisonofQSAR … · 2020. 3. 19. · Boscet al. J Cheminform Page3of16 Dta preparation Compoundstructureswereextractedfromthedatabase inSMILESformatandusingRDKit(version2017_09_01)

ZnO nanoparticles/silica for biginelli solution syntheisjournals.iau.ir/article_523134_d3e1e0618b5b13b0d2e... · [6]The Biginelli reaction, discovered by pietroBiginelli in 1893,

ZnO nanoparticles/silica for biginelli solution syntheisjournals.iau.ir/article_523134_d3e1e0618b5b13b0d2e... · [6]The Biginelli reaction, discovered by pietroBiginelli in 1893,

A mini-review on Biginelli adducts with notable ... the disclosure of Biginelli reaction by the chemist Pietro Biginelli, functionalized 3,4-dihy-dropyrimidin-2(1H)-ones/thiones (DHPMs)

A mini-review on Biginelli adducts with notable ... the disclosure of Biginelli reaction by the chemist Pietro Biginelli, functionalized 3,4-dihy-dropyrimidin-2(1H)-ones/thiones (DHPMs)

Conceptos fundamentales y preparación de expedientes ...echa.europa.eu/documents/10162/13566/uvcb_gabriele... · indeno/indano, naftaleno y homólogos, hidrocarburos nafténicos

Conceptos fundamentales y preparación de expedientes ...echa.europa.eu/documents/10162/13566/uvcb_gabriele... · indeno/indano, naftaleno y homólogos, hidrocarburos nafténicos

Ionic Liquid Effect over the Biginelli Reaction - Ainfo - Embrapa

Ionic Liquid Effect over the Biginelli Reaction - Ainfo - Embrapa

Polycyclic aromatic hydrocarbons (PAHs) concentration ...kjc.njfu.edu.cn/uploads/file/20180719/20180719105107_19706.pdf · indeno(1,2,3-cd)-pyrene (IcdP). In this study, the extracts

Polycyclic aromatic hydrocarbons (PAHs) concentration ...kjc.njfu.edu.cn/uploads/file/20180719/20180719105107_19706.pdf · indeno(1,2,3-cd)-pyrene (IcdP). In this study, the extracts

Classification System for Solid Supports Used ... - FIZ CHEMIE › fileadmin › user_upload › Cheminform › Spore › _… · FIZ CHEMIE BERLIN - 5 (23) - The remainder of the

Classification System for Solid Supports Used ... - FIZ CHEMIE › fileadmin › user_upload › Cheminform › Spore › _… · FIZ CHEMIE BERLIN - 5 (23) - The remainder of the

ChemInform RxnFinder

ChemInform RxnFinder

A new insight into the Biginelli reaction: the dawn of ... · PDF file1 Supporting Information A new insight into the Biginelli reaction: the dawn of multicomponent click chemistry?

A new insight into the Biginelli reaction: the dawn of ... · PDF file1 Supporting Information A new insight into the Biginelli reaction: the dawn of multicomponent click chemistry?

Laporan Percobaan Biginelli New

Laporan Percobaan Biginelli New

Synthesis of structurally diverse 3,4-dihydropyrimidin-2 ... · Synthesis of structurally diverse 3,4-dihydropyrimidin-2(1H)-ones via sequential Biginelli and Passerini reactions

Synthesis of structurally diverse 3,4-dihydropyrimidin-2 ... · Synthesis of structurally diverse 3,4-dihydropyrimidin-2(1H)-ones via sequential Biginelli and Passerini reactions

Hydrothermal Synthesis, Characterization and Catalytic ...jns.kashanu.ac.ir/article_87906_709df3439fd3da4a9b43ddc3771df776.pdfThe Biginelli reaction was originally reported by Biginelli

Hydrothermal Synthesis, Characterization and Catalytic ...jns.kashanu.ac.ir/article_87906_709df3439fd3da4a9b43ddc3771df776.pdfThe Biginelli reaction was originally reported by Biginelli

MATERIAL PARTICULADO EMITIDO EM … · Hidrocarbonetos policiclicos aromáticos Indeno( 1,2,3-cd)pireno ... analisados os alcanos e HPA presentes no material particulado de amostras

MATERIAL PARTICULADO EMITIDO EM … · Hidrocarbonetos policiclicos aromáticos Indeno( 1,2,3-cd)pireno ... analisados os alcanos e HPA presentes no material particulado de amostras

METHODOLOGY Molecularstructuresenumeration and ......Koch et al. J Cheminform Page5of17 changing4bonds,sinceweaimtondminimaltransfor - mations.Letuscall a 13 and a 24 thetwofixedbonds,with

METHODOLOGY Molecularstructuresenumeration and ......Koch et al. J Cheminform Page5of17 changing4bonds,sinceweaimtondminimaltransfor - mations.Letuscall a 13 and a 24 thetwofixedbonds,with

3,4— 二氢嘧啶酮的合成 ----Biginelli 反应

3,4— 二氢嘧啶酮的合成 ----Biginelli 反应

Español English Français - ACTA · indano indane indane. azul de indantrona indanthrone blue bleu d’indanthrène indazol indazole indazole indeno indene indène indio indium indium

Español English Français - ACTA · indano indane indane. azul de indantrona indanthrone blue bleu d’indanthrène indazol indazole indazole indeno indene indène indio indium indium