ChemInform Abstract: Synthesis and Biological Evaluation of Conduritol and Conduramine Analogues.

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1999 carbohydrates carbohydrates U 0500 30 - 209 Synthesis and Biological Evaluation of Conduritol and Conduramine Analogues. A number of conduritol and conduramine analogues are synthesized from naphthalene to give oxygenated derivatives with high stereo- and regiocontrol in a few steps. None of these compounds exhibit interesting enzymatic inhibitory activity against common glycosidases. (DESJARDINS, MICHEL; LALLEMAND, MARIE-CHRISTINE; FREEMAN, STANLEY; HUDLICKY, TOMAS; ABBOUD, KHALIL A.; J. Chem. Soc., Perkin Trans. 1 [old] (1999) 5, 621-628; Dep. Chem., Univ. Fla., Gainesville, FL 32611, USA; EN) 1

Transcript of ChemInform Abstract: Synthesis and Biological Evaluation of Conduritol and Conduramine Analogues.

Page 1: ChemInform Abstract: Synthesis and Biological Evaluation of Conduritol and Conduramine Analogues.

1999 carbohydrates

carbohydratesU 0500

30 - 209Synthesis and Biological Evaluation of Conduritol and ConduramineAnalogues. — A number of conduritol and conduramine analoguesare synthesized from naphthalene to give oxygenated derivatives with highstereo- and regiocontrol in a few steps. None of these compounds exhibitinteresting enzymatic inhibitory activity against common glycosidases. —(DESJARDINS, MICHEL; LALLEMAND, MARIE-CHRISTINE; FREEMAN,STANLEY; HUDLICKY, TOMAS; ABBOUD, KHALIL A.; J. Chem. Soc.,Perkin Trans. 1 [old] (1999) 5, 621-628; Dep. Chem., Univ. Fla., Gainesville,FL 32611, USA; EN)

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