2003-2004 Antineoplastics 1 February 2016 3:08 AM.
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Transcript of 2003-2004 Antineoplastics 1 February 2016 3:08 AM.
2003-2004Antineoplastics
May 3, 202306:01 PM
Alemtuzumab
Antineoplastic
Anti-CD52 antibody
Aminoglutethimide
AntineoplasticImmunosuppressive
Glucocorticoid antagonistAromatase inhibitor
(decreases steroid synthesis)
Amsacrine
Antineoplastic
Miscellaneous
Anastrozole
AntineoplasticAntiestrogen
Aromatase inhibitor
L-asparaginase
Antineoplastic
Protein synthesis inhibitor
Azathioprine
ImmunosuppressiveAntineoplastic
Antimetabolite(“pseudofeedback inhibition” of
HGPRT and PRP)
Bleomycin
Antineoplastic
Natural productAntibiotic
Busulfan
Antineoplastic
Alkylating Agent
Carmustine (BCNU)
Antineoplastic
Alkylating Agent
Cisplatin
Antineoplastic
MiscellaneousCross-linking agent
Cyclophosphamide
Antineoplastic
Alkylating Agent
Cyclosporine
ImmunosuppressiveAntineoplastic
Binds cyclophilinInhibits calcineurin
Cyproterone acetate
AntiandrogenAntineoplastic
androgen receptor antagonist
Cytarabine (AraC)
Antineoplastic
Antimetabolite
Dacarbazine
Antineoplastic
Alkylating Agent
Dactinomycin
Antineoplastic
Natural productAntibiotic
Daunorubicin
Antineoplastic
Anthracycline antibiotic Natural product
Dexamethasone
AdrenocorticosteroidGlucocorticoidAntineoplastic
Anti-inflammatory steroidNot by inhalation
Doxorubicin
Antineoplastic
Anthracycline antibioticNatural product
Etoposide
Antineoplastic
Natural productPlant alkaloid
Exemestane
AntineoplasticAntiestrogen
Aromatase Inhibitor
5-Fluorouracil
Antineoplastic
AntimetaboliteThymidylate synthase inhibitor
Fulvestrant
AntineoplasticAntiestrogen
Estrogen receptor antagonist
Gemtuzumab
Antineoplastic
Anti-CD33 antibody
Goserelin
AntineoplasticGonadotropin releasing
hormone(GnRH) agonist
Hydroxyurea
Antineoplastic
MiscellaneousRibonucleotide reductase
inhibitor
Ibritumomab
Antineoplastic
Anti-CD20 antibody
Imatinib
Antineoplastic
MiscellaneousTyrosine kinase inhibitor
Interleukin 2
Cytokine Antineoplastic
Interleukin 11
Cytokine Antineoplastic (supporting
agent)
Iressa
Antineoplastic
MiscellaneousTyrosine kinase inhibitor
Letrozole
AntineoplasticAntiestrogen
Aromatase Inhibitor
Leucovorin
Antineoplastic (supporting agent)
Folic acid analogue(used in methotrexate rescue)
Leuprolide
AntineoplasticGonadotropin releasing hormone (GnRH) agonist
Lomustine (CCNU)
Antineoplastic
Alkylating Agent
Mechlorethamine
Antineoplastic
Alkylating Agent
Melphalan
Antineoplastic
Alkylating Agent
6-Mercaptopurine
Antineoplastic
Antimetabolite(“pseudofeedback inhibition” of
HGPRT and PRP – purine synthesis)
Mesna
Antineoplastic (supporting agent)
Prevent hemorrhagic cystitisdue to cyclophosphamide
Methotrexate
ImmunosuppressiveAntineoplastic
Folic acid antagonistDihydrofolate reductase
inhibitor
Mitomycin C
Antineoplastic
Natural productAntibiotic
Paclitaxel
Antineoplastic
Natural productPlant alkaloid (taxane)
Pentostatin
Antineoplastic
MiscellaneousEnzyme inhibitor
(blocks purine synthesis)
Rituxumab
Antineoplastic
Anti-CD20 antibody
Tacrolimus
ImmunosuppressiveAntineoplastic
Binds FKBP (FK506 binding protein)
Inhibits calcineurin
Thalidomide
Antineoplastic
Anti-angiogenicAnti-TNF
Leprosy (not antibiotic)
6-Thioguanine
Antineoplastic
Antimetabolite (“pseudofeedback inhibition” of
HGPRT and PRP – purine synthesis)
Thiotepa
Antineoplastic
Alkylating agent
Trastuzumab
Antineoplastic
Anti-HER2 antibody
Tumor necrosis factor
CytokineAntineoplastic
Vinblastine
Antineoplastic
Vinca alkaloidNatural product
Vincristine
Antineoplastic
Vinca alkaloidNatural product